1.药物与血浆蛋白的结合( )A.是可逆的
2.量反应的量效曲线( )B.横坐标为药物对数浓度,纵坐标为药物的效应,呈对称的S形曲线
3.影响药物从体内排泄的因素不包括( )
C.药物剂量
4.促进药物生物转化的主要酶系统是( )B.细胞色素P-450酶系统
5.通过激动α受体产生的效应是( )D.瞳孔扩大
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6.治疗量阿托品不会引起( ) C.中枢兴奋,焦虑不安
阿托品竞争性拮抗ACh或胆碱受体激动药对M胆碱受体的激动作用。
7.不属于琥珀胆碱作用特点的是( )B.过量可引起呼吸麻痹
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8.肾上腺素对心脏的作用是( ) B.激动β1受体,使心率加快,心肌收缩力加强,传导加快
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9.异丙肾上腺素不具有的作用( ) D.收缩支气管粘膜血管
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10.酚妥拉明扩张血管的原因是( )B.阻断α受体
【药效学】本品为α—受体阻断剂。能显著降低外周血管阻力,增加血容量,增加组织血流量,改善微循环,改善内脏血流灌注,其作用比妥拉苏林强。
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11.治疗焦虑症最好选用( )B.地西泮
12.与苯二氮类药物比较,巴比妥类镇静催眠的缺点是( )D.抑制呼吸
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13.苯妥英钠的体内药物动力学的特点为( ) B.可静注和肌注给药
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14.左旋多巴治疗肝昏迷是由于( ) A.在脑内脱羧生成多巴胺
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15.由于长期应用氯丙嗪,使多巴胺受体上调而产生的副作用是( ) D.迟发性运动障碍
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16.有关吗啡的描述错误的是( ) D.抑制全身各种感觉,包括痛觉
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17.吗啡引起瞳孔缩小的机理是( ) D.激动中脑盖前核的阿片受体
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18.阿司匹林引起的凝血障碍可用何药预防( )A.鱼精蛋白
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9.对急性心肌梗塞引起的室性心动过速,首选( )D.利多卡因
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20.强心苷正性肌力作用的发生机制是( )B.抑制心肌细胞膜Na+,K+-ATP酶